• 11995 Citations
  • 54 h-Index
1974 …2018
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  • 7 Similar Profiles
Ligands Medicine & Life Sciences
Pharmacology Medicine & Life Sciences
Drug Discovery Medicine & Life Sciences
G-Protein-Coupled Receptors Medicine & Life Sciences
Drug Receptors Medicine & Life Sciences
Pharmaceutical Preparations Medicine & Life Sciences
GTP-Binding Proteins Medicine & Life Sciences
Adrenergic Receptors Medicine & Life Sciences

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Projects 2007 2017

Research Output 1974 2018

Is the quest for signaling bias worth the effort?

Kenakin, T. Apr 1 2018 In : Molecular pharmacology. 93, 4, p. 266-269 4 p.

Research output: Contribution to journalArticle

Health Expenditures
Drug Therapy
In Vitro Techniques

PAM-Antagonists: A Better Way to Block Pathological Receptor Signaling?

Kenakin, T. & Strachan, R. T. Jan 1 2018 (Accepted/In press) In : Trends in pharmacological sciences.

Research output: Contribution to journalArticle

7 Citations

Allosteric Modulation: An Alternate Approach Targeting the Cannabinoid CB1 Receptor

Nguyen, T., Li, J. X., Thomas, B. F., Wiley, J. L., Kenakin, T. P. & Zhang, Y. May 1 2017 In : Medicinal Research Reviews. 37, 3, p. 441-474 34 p.

Research output: Contribution to journalReview article

Cannabinoid Receptor CB1
Allosteric Site
Biological Phenomena

A new molecular mechanism to engineer protean agonism at a G protein-coupled receptor

De Min, A., Matera, C., Bock, A., Holze, J., Kloeckner, J., Muth, M., Traenkle, C., De Amici, M., Kenakin, T., Holzgrabe, U., Dallanoce, C., Kostenis, E., Mohr, K. & Schrage, R. Apr 1 2017 In : Molecular pharmacology. 91, 4, p. 348-356 9 p.

Research output: Contribution to journalArticle

G-Protein-Coupled Receptors
Cholinergic Receptors
Cholinergic Agents
Molecular Probes
2 Citations

A Scale of Agonism and Allosteric Modulation for Assessment of Selectivity, Bias, and Receptor Mutation

Kenakin, T. Oct 1 2017 In : Molecular pharmacology. 92, 4, p. 414-424 11 p.

Research output: Contribution to journalReview article

Drug Agonism
Drug Dose Response Relationship
Allosteric Regulation
Structure-Activity Relationship
Cytoplasmic and Nuclear Receptors